In Vitro Pharmacological Screening of Essential Oils from Baccharis parvidentata and Lippia origanoides Growing in Brazilстатья
Статья опубликована в журнале из списка Web of Science и/или Scopus
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Авторы:
Perera W.H.,
Scherbakov A.M.,
Buravchenko G.I.,
Mikhaevich E.I.,
Leitão S.G.,
Cos P.,
Shchekotikhin A.E.,
Monzote L.,
Setzer W.N.
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Журнал:
Molecules
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Том:
27
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Номер:
6
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Год издания:
2022
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Издательство:
MDPI
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Местоположение издательства:
Basel, Switzerland
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DOI:
10.3390/molecules27061926
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Аннотация:
In this study, the in vitro antimicrobial, antiparasitic, antiproliferative and cytotoxic activities of essential oil from Baccharis parvidentata Malag. (EO-Bp) and Lippia origanoides Kunth (EO-Lo) were explored. The relevant effects were observed against the parasitic protozoans Plasmodium falciparum, Trypanosoma cruzi, Trypanosoma brucei and Leishmania amazonensis (ranging 0.6 to 39.7 µg/mL) and malignant MCF-7, MCF-7/HT, 22Rv1, and A431 cell lines (ranging 6.1 to 31.5 µg/mL). In parallel, EO-Bp showed better selective indexes in comparison with EO-Lo against peritoneal macrophages from BALB/c mice and MRC-5 cell line. In conclusion, EO-Lo is known to show a wide range of health benefits that could be added as another potential use of this oil with the current study. In the case of EO-Bp, the wide spectrum of its activities against protozoal parasites and malignant cells, as well as its selectivity in comparison with non-malignant cells, could suggest an interesting candidate for further tests as a new therapeutic alternative. © 2022 by the authors. Licensee MDPI, Basel, Switzerland.
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Добавил в систему:
Малошицкая Ольга Александровна